Saturday, July 22, 2017

Game of precursors




Why nad+?

It is part of the inner chargeable battery that cycles between nad+ and nadh.
Why not synthesize nadh directly?

There are no direct reactions of substance. Only nad+ can be increased, in turn food will charge it to increased nadh. Mind you, the energy recovery is by unit weight. So either nadh or nad+ has to be synthesized

Why increase nad+ by nature way?

At this point, nature is mimicked. Someday, some bio scientist-engineers will claim other ways of synthesis and their methods will have centuries of anti-cancer testing. Till then, the conservative safe way is to mimic nature!

How increase nad+ by nature way?

We can do it by examining the precursors in various organic reactions.  Also one must consider the amount delivered. We have to cross the stomach-blood barrier and then the chemical has to be ingested by the cell. Collectively we call the crossing the bioavailability.

Why hard?

The cheapest way to increase calcium is to eat chalk. Bad idea because the chemical may damage the stomach and has negligible bioavailability. Same is not true of some complex bio-molecules with Ca ion. Even the best have maximal absorption rates, so there is NO instantaneous way of raising!

How come you know re Ca?

My mother has been diagnosed deficient in Ca, fundamental cause of osteoporosis. Interesting ways to increase Ca makes sense to me!

How can you improve bioavailability of anything?

No matter what it is, element  ion or salt, you can always inject it into the blood stream directly. Problem is you bypass the stomach-blood filter that performs two essentials – keep out the impurities and convert it right blood form. It means that injectable be medical-grade pure and known to be injectable! An anti-oxidant Glutathione which also disrupts melanin synthesis has this property and slowly, doctors are opening direct-IV centers that advertise proven Skin-whitening for girl-marriage with guaranteed whitening for a few months.

Precursors?

There are many to nad+. They require 2 or more steps to become nad+. Further away you are, lower the effectiveness because of increased bio-availability issues and increased chances of unintended side effects. All start with vitamin B3, most have similar pathways to nad+ and similar bad side-effect profile – in other words safe to high doses . This makes them perfect  goods for semi-intelligents to be thugged in honest ways. Point is these are all precursors, they can each do the job, may or may not in reality, discovery is incredible hard, there are plenty of anecdotal-advice givers and wise-oracles buyable. In other words, intellectual debates best avoided. What can clear the nonsense are high quality studies, started for niagen in Japan and metformin in USA, but due in 2020. Even the need for such studies are a positive sign beyond amazon hype!

NR?

Nam, Na, and Trp (Tryptophan) are advertised, sold but shown ineffective precursors to nad+. Note that even earlier is B3 (niacin) in two forms, dangerous flushing niacin and non-flushing niacinamide. Another approach to non-flushing is time-release version of niacin. All these are as far away as B3 (First N in most is niacin). Much closer (closest) is NR. The riboside molecule seems to have better bio-availability for most in conjunction with exercise (I posit). Note that NR might be essential to motivate oldies  to exercise some, in the first place (past the feeling of enervation!). It is a good place to bet because Japanese are at least studying it! Best not bet but wait till 2018, but only if you can. It is NOT a shame to fall for amazon hype,  perhaps. At worst, very good chances are you wasted money at most.

Metformin?

CDC in USA studies it. Even more specialized studies operate. Early mother of investigations was a statistical study from 2000 + in UK that compared lifespans of metformin alone treated diabetics M, equivalent free of diabetes F and equivalent  insulin treated diabetics I; and found N – 5 > F > I + 5. Eating metformin seems to do the trick unless equivalency used by statisticians was bullshit! Started the study in 2016. A Swedish study pph-poohed renal damage, stating - Conclusions Metformin showed lower risk than insulin for CVD and all-cause mortality and slightly lower risk for all-cause mortality compared with other OHA, in these 51 675 patients followed for 4 years. Patients with renal impairment showed no increased risk of CVD, all-cause mortality or acidosis/serious infection. In clinical practice, the benefits of metformin use clearly outbalance the risk of severe side effects.
 How evil is sugars? VERY.

The United Kingdom Prospective Diabetes Study (UKPDS) set out to examine the effect of intensified glucose control upon the subsequent development of complications of diabetes in newly diagnosed patients, and the relative benefits of specific therapies (diet, sulfonylureas, metformin or insulin) in this regard. It recruited 5,102 patients from 23 centres between 1977 and 1991. Patients were followed for an average of 10 years. A blood pressure arm was added in the course of the study and compared rigorous vs less rigorous blood pressure control in hypertensive people with diabetes, and the relative benefits of an ACE inhibitor (captopril) or β-blocker (atenolol) in achieving this. Median HbA1c was 7.9% on conventional therapy and 7.0% on intensified therapy, and this was associated with a 25% reduction in the rates of retinopathy, nephropathy and (possibly) neuropathy. Results were even stronger in the epidemiological arm (which compared achieved HbA1c rather than treatment arm), and no glycaemic threshold for complications was observed. There was a non-significant 16% reduction in myocardial infarction or sudden death with intensified therapy, and a 25% reduction in the risk of death for every 1% drop in HbA1c. Antihypertensive therapy markedly reduced all end-points, microvascular as well as arterial.


WARNING: I AM no DOCTOR, nor are you. Get encouraged to visit and not appear stupid

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